您的位置：首页 > 产品中心 > 189188-57-6， Tegaserod maleate
Tegaserod maleate
产品别名
189188-57-6
Tegaserod maleate
2-[(5-Methoxy-1H-indol-3-yl)methylene]-N-pentyl-hydrazinecarboximidamide maleate
结构式
基本信息
| Empirical Formula【经验(实验)分子式】 | C16H23N5O · C4H4O4 |
| Molecular weight | 417.46 |
| MDL number | MFCD09028009 |
| PubChem Substance ID【PubChem化学物质编号】 | 329825925 |
| NACRES | NA.77 |
| Application【应用】 | Tegaserod maleate has been used to study its cytotoxic effects on human astrocytes and to study its effects as an anti-glioblastoma agent. |
| Biochem/physiol Actions【生化/生理作用】 | It stimulates neurotransmitter release from enteric nerves and regularizes gastrointestinal function. Tegaserod has been used to treat irritable bowel syndrome associated with constipation and chronic constipation. Tegaserod is a potent full agonist at serotonin 5-HT4 receptors with an EC50 of 7 nM. |
产品性质
| Quality Level【质量水平】 | 100 |
| Assay【测定】 | ≥98% (HPLC) |
| form【形式】 | powder |
| color【颜色】 | white to beige |
| solubility【溶解性】 | DMSO: 20 mg/mL, clear |
| storage temp.【储存温度】 | 2-8℃ |
| SMILES string | N=C(NCCCCC)N/N=C/C1=CNC2=C1C=C(OC)C=C2.OC(/C=C\C(O)=O)=O |
| InChI | 1S/C16H23N5O.C4H4O4/c1-3-4-5-8-18-16(17)21-20-11-12-10-19-15-7-6-13(22-2)9-14(12)15;5-3(6)1-2-4(7)8/h6-7,9-11,19H,3-5,8H2,1-2H3,(H3,17,18,21);1-2H,(H,5,6)(H,7,8)/b20-11+;2-1- |
| InChI key | CPDDZSSEAVLMRY-FEQFWAPWSA-N |
| Gene Information | human ... HTR4(3360) |
| packaging【包装】 | 10, 50 mg in glass bottle |
安全信息
| Storage Class Code【储存分类代码】 | 13 - Non Combustible Solids |
| WGK | WGK 3 |
