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GP Antagonist-2A-Calbiochem
| 产品编号： | 4061839 |
| 规格： | The GP Antagonist-2A controls the biological activity of GP. This small molecule/inhibitor is primarily used for Neuroscience applications. |
| 包装规格： | 1 MG |
| 产品类别： | 进口试剂 |
| 品牌： | Sigma-Aldrich |
| 优惠价： | 立即咨询 |
产品别名
GP Antagonist-2A-Calbiochem
RPKPQQDWFDWDWM
基本信息
| Empirical Formula【经验(实验)分子式】 | C79H105N21O13S |
| Molecular weight | 1588.88 |
| General description【一般描述】 | A peptide that selectively inhibits the activation of Gq by M1-muscarinic cholinergic receptors. Also inhibits activation by cholecystokinin receptor in pancreatic acini at 10 µM. Blocks angiotensin II-stimulated sis-inducing factor and STAT3 tyrosine phosphorylation. |
| Biochem/physiol Actions【生化/生理作用】 | Product does not compete with ATP. Reversible: no Primary Target Inhibits the activation of Gq by M1-muscarinic cholinergic receptors Cell permeable: no |
| Warning【警告】 | Toxicity: Standard Handling (A) |
| Sequence【序列】 | H-Arg-Pro-Lys-Pro-Gln-Gln-D-Trp-Phe-D-Trp-D-Trp-Met-NH₂ |
| Other Notes【其他说明】 | Hunt, R.A., et al. 1999. Hypertension34, 603. Tsunoda Y., et al. 1995. Biochem. Biophys. Res. Commun. 211, 648. Mukai, H., et al. 1992. J. Biol. Chem.267, 16237. |
| Legal Information【法律信息】 | CALBIOCHEM is a registered trademark of Merck KGaA, Darmstadt, Germany |
产品性质
| Quality Level【质量水平】 | 100 |
| Assay【测定】 | ≥95% (HPLC) |
| form【形式】 | lyophilized solid |
| manufacturer/tradename | Calbiochem® |
| storage condition【储存条件】 | OK to freeze |
| solubility【溶解性】 | water: 25 mg/mL |
| shipped in【运输】 | ambient |
| storage temp.【储存温度】 | −20℃ |
| packaging【包装】 | 1 mg in Plastic ampoule |
安全信息
| Storage Class Code【储存分类代码】 | 11 - Combustible Solids |
| WGK | WGK 1 |
