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产品别名
BQ-788, Sodium Salt-CAS-Calbiochem
N- cis-2,6-Dimethylpiperidinocarbonyl-L-γ-MeLeu-D-Trp(MeOCO)-D-Nle-OH, Na
基本信息
| Empirical Formula【经验(实验)分子式】 | C34H50N5NaO7 |
| Molecular weight | 663.78 |
| General description【一般描述】 | A highly selective and competitive ETB receptor antagonist (IC50 = 1.2 nM). Highly selective ETB-receptor antagonist (IC50 = 1.2 nM). |
| Biochem/physiol Actions【生化/生理作用】 | Primary Target ETB-receptor antagonist Target IC50: 1.2 nM as ETB-receptor antagonist Product does not compete with ATP. Reversible: no Cell permeable: no |
| Warning【警告】 | Toxicity: Standard Handling (A) |
| Reconstitution【重悬】 | Following reconstitution, aliquot and freeze (-20°C). DMSO and Methano:H₂O stock solutions are stable for up to 2 months at -20°C. |
| Other Notes【其他说明】 | Okada, M., and Nishikibe, M. 2002. Cardiovasc. Drug Reviews20, 53. Taniai, H., et al. 2001. Hepatology33, 894. Fukuroda, T., et al. 1994. Biochem. Biophys. Res. Commun.199, 1461. Ishikawa, K., et al. 1994. Proc. Natl. Acad. Sci. USA91, 4892. |
| Legal Information【法律信息】 | CALBIOCHEM is a registered trademark of Merck KGaA, Darmstadt, Germany |
产品性质
| Quality Level【质量水平】 | 100 |
| Assay【测定】 | ≥95% (HPLC) |
| form【形式】 | lyophilized solid |
| manufacturer/tradename | Calbiochem® |
| storage condition【储存条件】 | OK to freeze desiccated |
| color【颜色】 | white to off-white |
| solubility【溶解性】 | 0.01% NH4OH: 1 mg/mL DMSO: 2 mg/mL methanol: water (3:1): 2 mg/mL |
| shipped in【运输】 | ambient |
| storage temp.【储存温度】 | −20℃ |
安全信息
| Storage Class Code【储存分类代码】 | 11 - Combustible Solids |
| WGK | WGK 1 |
