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VPC-13566
产品别名
218464-59-6
VPC-13566
2-(7-Methyl-1H-indol-3-yl)quinoline
结构式
基本信息
| Empirical Formula【经验(实验)分子式】 | C18H14N2 |
| Molecular weight | 258.32 |
| NACRES | NA.77 |
| Biochem/physiol Actions【生化/生理作用】 | VPC-13566 is Binding Function 3 (BF3)-specific inhibitor of the androgen receptor. VPC-13566 potently inhibits AR transcriptional activity by displacement of the BAG1L peptide from the BF3 pocket. VPC-13566 inhibits the growth of various prostate cancer cell lines including an enzalutamide-resistant cell line and inhibits the growth of AR-dependent prostate cancer xenograft in mice. |
产品性质
| Quality Level【质量水平】 | 100 |
| Assay【测定】 | ≥98% (HPLC) |
| form【形式】 | powder |
| color【颜色】 | white to beige |
| solubility【溶解性】 | DMSO: 20 mg/mL, clear |
| storage temp.【储存温度】 | 2-8℃ |
| SMILES string | CC1=CC=CC2=C1NC=C2C3=NC4=CC=CC=C4C=C3 |
| packaging【包装】 | 5, 25 mg in glass bottle |
安全信息
| Storage Class Code【储存分类代码】 | 13 - Non Combustible Solids |
| WGK | WGK 3 |
