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PKC Inhibitor, EGF-R Fragment 651-658, Myristoylated-Calbiochem
| 产品编号： | 4146279 |
| 规格： | The PKC Inhibitor, EGF-R Fragment 651-658, Myristoylated controls the biological activity of PKC. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications. |
| 包装规格： | 500 μG |
| 产品类别： | 进口试剂 |
| 品牌： | Sigma-Aldrich |
| 优惠价： | 立即咨询 |
产品别名
PKC Inhibitor, EGF-R Fragment 651-658, Myristoylated-Calbiochem
Myr-N-RKRTLRRL-OH, Myristoylated EGF-R Fragment (651-658), Protein Kinase C Inhibitor, Protein Kinase C Inhibitor, EGF-R Fragment 651-658, Myristoylated
Myristoylated EGF-R Fragment (651-658), Protein Kinase C Inhibitor, Myr-N-RKRTLRRL-OH, Protein Kinase C Inhibitor, EGF-R Fragment 651-658, Myristoylated
基本信息
| Empirical Formula【经验(实验)分子式】 | C60H117N21O11 |
| Molecular weight | 1308.71 |
| General description【一般描述】 | Epidermal growth-factor receptor (EGF-R) conserved sequence which is identical to v-erbB (95-102). An N-terminal myristoylated membrane-permeable, reversible, and substrate competitive inhibitor that inhibits protein kinase C (IC50 = 5 µM) in intact cells. Epidermal growth-factor receptor (EGF-R) conserved sequence which is identical to v-ErbB (95-102). An N-terminal myristoylated membrane-permeable, reversible, and substrate competitive inhibitor of protein kinase C (IC50 = 5 µM). |
| Biochem/physiol Actions【生化/生理作用】 | Product does not compete with ATP. Target IC50: 5 µM against protein kinase C Reversible: yes Primary Target PKC Cell permeable: yes |
| Warning【警告】 | Toxicity: Standard Handling (A) |
| Sequence【序列】 | Myr-N-Arg-Lys-Arg-Thr-Leu-Arg-Arg-Leu-OH |
| Physical form【外形】 | Supplied as a trifluoroacetate salt. |
| Reconstitution【重悬】 | Following reconstitution, aliquot and freeze (-20°C). Stock solutions are stable for up to 2 months at -20°C. |
| Other Notes【其他说明】 | Ward, N.E., and O’Brian, C.A. 1993. Biochemistry32, 11903. O’Brian, C.A., et al. 1991. Invest. New Drugs 9, 169. |
| Legal Information【法律信息】 | CALBIOCHEM is a registered trademark of Merck KGaA, Darmstadt, Germany |
产品性质
| Quality Level【质量水平】 | 100 |
| Assay【测定】 | ≥97% (HPLC) |
| form【形式】 | lyophilized solid |
| manufacturer/tradename | Calbiochem® |
| storage condition【储存条件】 | OK to freeze desiccated |
| solubility【溶解性】 | water: 5 mg/mL |
| shipped in【运输】 | ambient |
| storage temp.【储存温度】 | −20℃ |
| packaging【包装】 | 500 μg in Plastic ampoule Yes |
安全信息
| Storage Class Code【储存分类代码】 | 11 - Combustible Solids |
| WGK | WGK 1 |
