产品编号：4083741

纯度规格：A cell permeable, selective, sphingosine competitive inhibitor of spingosine Kinase -2 (IC₅₀ = 4.3 μM).

包装规格：10 MG

产品编号：4083740

纯度规格：A peptidyl toxin from venom of African tarantula, Hysterocrates gigas that acts as a high affinity, reversible blocker of Cav2.3 (α1E, R-type) channels (IC₅₀ = 15-30 nM).

包装规格：10 μG

产品编号：4083738

纯度规格：A cell-permeable inhibitor of SKP2-dependent p27Kip1 ubiquitination. Selectively induces the accumulation SCFSKP2 substrates in multiple myeloma RPMI 8226 cells.

包装规格：10 MG

产品编号：4083737

包装规格：10 MG

产品编号：4083736

纯度规格：A highly potent agonist of GABAB receptor. Shown to be about 10-times more potent than baclofen.

包装规格：10 MG

产品编号：4083734

包装规格：10 MG

产品编号：4083725

纯度规格：A cell-permeable racemic mixture of Halofuginone that inhibits of prolyl-tRNA synthetase.

包装规格：10 MG

产品编号：4083724

纯度规格：A cell-permeable, selective inhibitor of protein arginine methyltransferase 1 (PRMT1; IC₅₀ = 9.5 μM).

包装规格：10 MG

产品编号：4083722

包装规格：10 MG

产品编号：4083721

纯度规格：A cell-permeable inhibitor of Wnt secretion from L-cell Wnt1/2/3/3a/6/7a/9a transfectants (IC₅₀ from 50 pM to 1.1 nM).

包装规格：5 MG

产品编号：4083717

纯度规格：A rhodanine-derived, reversible, photoactivated, TrpA1-selective channel activator.

包装规格：10 MG

产品编号：4083714

纯度规格：A cell-permeable, highly potent and selective inhibitor of phosphodiesterase 5 (PDEV; IC₅₀ = 270 pM).

包装规格：5 MG

产品编号：4083710

纯度规格：A cell-permeable compound that selectively downregulates the expression of p21 (~10 μM), independent of p53.expression, at either transcription or post-transcriptional level.

包装规格：10 MG

产品编号：4083706

纯度规格：A cell-permeable myristoylated hexapeptide that selectively inhibits integrin outside-in signaling without affecting inside-out signaling. Blocks the interaction of Gα3 and integrin β3 subunit.

包装规格：10 MG

产品编号：4083701

纯度规格：A cell-permeable. Reversible, selective inhibitor of the growth of malignant peripheral nerve sheath tumors (EC₅₀ = 439 nM, 754 nM, and 1.0 μM in S462, SNF96.2, and sMPNST cells).

包装规格：25 MG

产品编号：4083697

包装规格：10 MG

产品编号：4083692

纯度规格：A cell-permeable, potent, selective, reversible inhibitor of Lysine-Specific Demethylase 1 (LSD1; IC₅₀ = 13 nM; K_i = 31 nM).

包装规格：10 MG

产品编号：4083691

纯度规格：A cell-permeable, both NADH and pyruvate-competitive isoform A-selective LDH inhibitor. Exhibits enhanced anticancer activity under hypoxic conditions.

包装规格：10 MG

产品编号：4083690

纯度规格：A cell-permeable, fast acting, branched polyamine. Induces growth of actin-enriched lamellipodia within minutes without the need for serum cofactors .

包装规格：10 MG

产品编号：4083688

纯度规格：A voltage gated calcium channel gating inhibitor of the dihydropyridine class.

包装规格：10 MG

产品编号：4083686

纯度规格：A substrate competitive inhibitor of insulin-regulated aminopeptidase (IRAP) activity (K_i = 0.48 μM against 25 μM Leu-AMC).

包装规格：10 MG

产品编号：4083685

纯度规格：A 10 mM (5 mg/1.07 ml) sterile-filtered solution of Wnt Antagonist II, IWP-2) in DMSO.

包装规格：5 MG

产品编号：4083683

纯度规格：A 25 mM (5 mg/357 μl) sterile-filtered solution of PPACK, 2HCl in H₂O.

包装规格：5 MG

产品编号：4083680

包装规格：10 MG

产品编号：4083678

纯度规格：A 50 mM sterile-filtered solution of I-BET in DMSO.

包装规格：5 MG

产品编号：4083677

纯度规格：A 25 mM (2 mg/231 μl) sterile-filtered solution of Ginkgolic Acid (15:1) in DMSO.

包装规格：2 MG

产品编号：4083676

包装规格：5 MG

产品编号：4083675

包装规格：2 MG

产品编号：4083674

纯度规格：A 25 mM solution of (+)-Brefeldin A in DMSO.

包装规格：2 MG

产品编号：4083672

纯度规格：A cell-permeable compound that competitively binds to Hu antigen R (HuR; K_i = 350 nM) and disrupts the interaction of HuR and adenine- and uridine-rich element (ARE) of target mRNAs.

包装规格：10 MG

产品编号：4083670

包装规格：10 MG

产品编号：4083667

纯度规格：Cell-permeable inhibitor of gp130. Binds to gp130 and induces its phosphorylation at Ser782 in ovarian cancer cells. Suppresses constitutive phosphorylation of and nuclear translocation of Stat3.

包装规格：10 MG

产品编号：4083664

产品编号：4083662

纯度规格：Specifically binds to the Fn14 surface (Kd = 7.12 mM) and suppresses TWEAK-induced glioma cell migration.

包装规格：10 MG

产品编号：4083661

纯度规格：A cell-permeable structural analog of E1 that acts as an equipotent, SAM-competitive inhibitor of Ezh2/PRC2 inhibitor (K_i = 0.5 to 3 nM against wt &mutant Ezh2-containing PRC2).

包装规格：5 MG

产品编号：4083658

包装规格：10 MG

产品编号：4083655

纯度规格：DHODH Inhibitor, DSM1, is a highly potent, competitive, tight-binding inhibitor of Plasmodium falciparum dihydroorotate dehydrogenase (IC₅₀ = 47 nM; K_i = 15 nM).

包装规格：25 MG

产品编号：4083653

包装规格：5 MG

产品编号：4083650

包装规格：10 MG

产品编号：4083649

包装规格：10 MG

产品编号：4083648

纯度规格：A 25 mM (10 mg/608 μL) sterile-filtered solution of CMP-Sialic Acid, Disodium Salt in H₂O.

包装规格：10 MG

产品编号：4083647

包装规格：25 MG

产品编号：4083645

纯度规格：A cell-permeable, highly potent, and specific inhibitor of CDC-like kinase (CLK; IC₅₀ = 1.1 and 2.4 nM for CLK1 and CLK2, respectively).

包装规格：5 MG

产品编号：4083644

纯度规格：A cell-permeable, potent, irreversible, non-substrate competitive inhibitor of CD45/PTPRC tyrosine phosphatase activity (IC₅₀ = 290 nM).

包装规格：10 MG

产品编号：4083642

纯度规格：Enhances BMP-2 associated signaling by inhibiting Smurf1-mediated Smad1/5 ubiquitination and thereby prolonging the half-life of Smad1 and 5. in 48 h).

包装规格：10 MG

产品编号：4083641

纯度规格：A cell-permeable compound that downregulates cellular BMI-1 levels by inhibiting BMI-1 transcription.

包装规格：10 MG

产品编号：4083640

纯度规格：A cell permeable, highly potent, selective inhibitor of Aurora A (IC₅₀ = 48 nM). Disrupts MYCN-Aurora A complex.

包装规格：10 MG

产品编号：4083638

纯度规格：A cell-permeable compound that directly and reversibly interacts with miRNA binding domain of Argonaute-2 (K_d = 126 μM) and inhibits binding of miR-20a, miR-26a, miR-107, miR-223 &let-7a to Ago2.

包装规格：25 MG

产品编号：4083634

纯度规格：Acid Ceramidase Inhibitor, BOC, CAS 1644158-57-5, is a cell-permeable, potent inhibitor of acid ceramidase (IC₅₀ = 79 nM against HEK293 lysosomal lysate AC activity).

包装规格：10 MG

产品编号：4083632

纯度规格：An anti-bacterial compound that targets NAD(P)H-dependent enoyl acyl carrier protein reductase (ENR) resulting in the inhibition of bacterial fatty acid synthase.

包装规格：10 MG